A One-pot Process For Preparation Of 2-substituted-1H-benzo[d]imidazole Derivatives
NIPER Raebareli
Chemical Sciences
Patent No. :
557854
Filed :
28-06-2024
Published :
13-01-2025
Granted
(E)-1-(2-(4-substituedphenyl)-2-oxoethyl)-4-((hydroxyimino)methyl)pyridinium bromides as anti-tubercular agents
KFU
Chemical Sciences
Patent No. :
US patent Pub No: US 12, 215, 082 B1
Filed :
26-06-2024
Published :
04-02-2025
Granted
A PROCESS FOR SYNTHESIS OF CHROMONE AND FLAVONE AND THEIR USE IN PHARMACEUTICAL APPLICATIONS
NIPER Raebareli
Chemical Sciences
Patent No. :
557480
Filed :
30-03-2024
Published :
06-01-2025
Granted
A PROCESS FOR SYNTHESIS OF CHROMONE AND FLAVONE AND THEIR USE IN PHARMACEUTICAL APPLICATIONS
NIPER Raebareli
Chemical Sciences
Patent No. :
557480
Filed :
30-03-2024
Published :
06-01-2025
Granted
A PROCESS FOR SYNTHESIS OF CHROMONE AND FLAVONE AND THEIR USE IN PHARMACEUTICAL APPLICATIONS
NIPER Raebareli
Chemical Sciences
Patent No. :
557480
Filed :
30-03-2024
Published :
06-01-2025
Granted
A PROCESS FOR SYNTHESIS OF CHROMONE AND FLAVONE AND THEIR USE IN PHARMACEUTICAL APPLICATIONS
NIPER Raebareli
Chemical Sciences
Patent No. :
557480
Filed :
30-03-2024
Published :
06-01-2025
Granted
Novel benzofuro[2,3-c]pyridinol compounds and process for preparation thereof
NIPER Raebareli
Chemical Sciences
Patent No. :
569870
Filed :
19-03-2024
Published :
19-08-2025
Granted
A PROCESS FOR PREPARATION OF BENZOFURAN AND BENZOFURO[2,3-C]PYRIDINE COMPOUNDS
NIPER Raebareli
Chemical Sciences
Patent No. :
552392
Filed :
11-03-2024
Published :
15-10-2024
Granted
Pyrrolo[1,2-a] imidazole, 1H-Pyrrole-3-carboxylate analogues and process for preparation thereof
NIPER Raebareli
Chemical Sciences
Patent No. :
553787
Filed :
21-02-2024
Published :
01-11-2024
Granted
Development of (E)-3-(substitutedbenzoyl)-7-((hydroxyimino)methyl)-2-substitutedindolizine-1-carboxylate derivatives as anti-tubercular agents
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Melendran Pillay
Pran Kishore Deb
Rashmi Venugopala
Viresh Mohanlall
Chemical Sciences
Application No. :
18/531,129
Filed :
06-12-2023
Published :
N/A
Filed
Development of (E)-3-(substitutedbenzoyl)-7-((hydroxyimino)methyl)-2-substitutedindolizine-1-carboxylate derivatives as anti-tubercular agents
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Melendran Pillay
Pran Kishore Deb
Rashmi Venugopala
Viresh Mohanlall
Chemical Sciences
Application No. :
18/531,129
Filed :
06-12-2023
Published :
N/A
Filed
(E)-1-(2-(4-substituedphenyl)-2-oxoethyl)-4-((hydroxyimino)methyl)pyridinium bromides as anti-tubercular agents.
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Melendran Pillay
Pran Kishore Deb
Rashmi Venugopala
Chemical Sciences
Application No. :
18386017
Filed :
23-11-2023
Published :
N/A
Filed
(E)-1-(2-(4-substituedphenyl)-2-oxoethyl)-4-((hydroxyimino)methyl)pyridinium bromides as anti-tubercular agents.
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Melendran Pillay
Pran Kishore Deb
Rashmi Venugopala
Chemical Sciences
Application No. :
18386017
Filed :
23-11-2023
Published :
N/A
Filed
Adenosine receptor activity of substituted benzoyl-7-methoxyindolizine-1-carboxylate analogues
Katharigatta N. Venugopala
Rahul D. Nagdeve
Pran Kishore Deb
Buccioni Michela
Gabriella Marucci
Susanta K. Nayak
Sandeep Chandrashekharappa
Osama I. Alwassil
Rashmi Venugopala
Chemical Sciences
Application No. :
18386397
Filed :
02-11-2023
Published :
N/A
Filed
Adenosine receptor activity of substituted benzoyl-7-methoxyindolizine-1-carboxylate analogues
Katharigatta N. Venugopala
Rahul D. Nagdeve
Pran Kishore Deb
Buccioni Michela
Gabriella Marucci
Susanta K. Nayak
Sandeep Chandrashekharappa
Osama I. Alwassil
Rashmi Venugopala
Chemical Sciences
Application No. :
18386397
Filed :
02-11-2023
Published :
N/A
Filed
7-Isopropyl 1-ethyl/methyl 3-(substituted benzoyl)-2-substituted indolizine-1,7-dicarboxylates as larvicidal agents
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Pran Kishore Deb
Osama I. Alwassil
Rashmi Venugopala.
Chemical Sciences
Application No. :
18/500,084,
Filed :
01-11-2023
Published :
N/A
Filed
7-Isopropyl 1-ethyl/methyl 3-(substituted benzoyl)-2-substituted indolizine-1,7-dicarboxylates as larvicidal agents
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Pran Kishore Deb
Osama I. Alwassil
Rashmi Venugopala.
Chemical Sciences
Application No. :
18/500,084,
Filed :
01-11-2023
Published :
N/A
Filed
4-Cyano-1-(2-oxo-2-(substituted phenyl)ethyl)pyridin-1-ium bromides as anti-tubercular agents.
Katharigatta N. Venugopala
Mohamed A. Morsy
Sandeep Chandrashekharappa
Melendran Pillay
Chemical Sciences
Application No. :
18384003
Filed :
26-10-2023
Published :
N/A
Filed
Ethyl-1-(substitutedbenzoyl)-5-methylpyrrolo[1,2-a]quinoline-3-carboxylates as anticancer agents
41. Katharigatta N. Venugopala
Vijaykumar Uppar
Rashmi Venugopala
Sandeep Chandrashekharappa
Basavaraj Padmashali
Chemical Sciences
Application No. :
18383407
Filed :
24-10-2023
Published :
N/A
Filed
Ethyl-1-(substitutedbenzoyl)-5-methylpyrrolo[1,2-a]quinoline-3-carboxylates as anticancer agents
41. Katharigatta N. Venugopala
Vijaykumar Uppar
Rashmi Venugopala
Sandeep Chandrashekharappa
Basavaraj Padmashali
Chemical Sciences
Application No. :
18383407
Filed :
24-10-2023
Published :
N/A
Filed
Substituted 7-amino-3-(substituted benzoyl)indolizine-1-carboxylates as anti-tubercular agents.
Katharigatta N. Venugopala
Melendran Pillay
Vijaykumar Uppar
Pran Kishore Deb
Rashmi Venugopala
Sandeep Chandrashekharappa
Basavaraj Padmashali
Chemical Sciences
Application No. :
18382829
Filed :
23-10-2023
Published :
N/A
Filed
Substituted 7-amino-3-(substituted benzoyl)indolizine-1-carboxylates as anti-tubercular agents.
Katharigatta N. Venugopala
Melendran Pillay
Vijaykumar Uppar
Pran Kishore Deb
Rashmi Venugopala
Sandeep Chandrashekharappa
Basavaraj Padmashali
Chemical Sciences
Application No. :
18382829
Filed :
23-10-2023
Published :
N/A
Filed
Ethyl-1-(substitutedbenzoyl)-5-methylpyrrolo [1, 2-a] quinoline-3-carboxylates as anticancer agents
Katharigatta N. Venugopala
Vijaykumar Uppar
Rashmi Venugopala
Sandeep Chandrashekharappa
Basavaraj Padmashali
Viresh Mohanlall.
Chemical Sciences
Patent No. :
US Patent 12,194,029,
Filed :
23-10-2023
Published :
14-01-2025
Granted
4-Cyano-1-(2-oxo-2-(substituted phenyl)ethyl)pyridin-1-ium bromides as anti-tubercular agents
Katharigatta N. Venugopala
Mohamed A. Morsy
Sandeep Chandrashekharappa
Melendran Pillay.
Chemical Sciences
Patent No. :
US 12, 202, 801 B1
Filed :
23-10-2023
Published :
21-01-2025
Granted
-(2-(SUBSTITUTED PHENYL)-2- OXOE- THYL)- 4-METHYLPYRIDIN-1-IUM BRO- MIDE AS ANTI-TUBERCULAR AGENTS
KFU
-
Patent No. :
US 12, 227, 480 B1
Filed :
23-10-2023
Published :
18-02-2025
Granted
Production of 1-(2-(substituted phenyl)-2-oxoethyl)-4-(isopropoxycarbonyl)pyridin-1-ium bromides and their anti-tubercular activity.
Katharigatta N. Venugopala
Pran Kishore Deb
Mohamed A. Morsy
Bandar E. Aldhubiab
Sandeep Chandrashekharappa
Melendran Pillay.
Chemical Sciences
Application No. :
Production of 1-(2-(substituted phenyl)-2-oxoethyl)-4-(isopropoxycarbonyl)pyridin-1-ium br
Filed :
10-10-2023
Published :
N/A
Filed
Production of 1-(2-(substituted phenyl)-2-oxoethyl)-4-(isopropoxycarbonyl)pyridin-1-ium bromides and their anti-tubercular activity.
Katharigatta N. Venugopala
Pran Kishore Deb
Mohamed A. Morsy
Bandar E. Aldhubiab
Sandeep Chandrashekharappa
Melendran Pillay.
Chemical Sciences
Application No. :
Production of 1-(2-(substituted phenyl)-2-oxoethyl)-4-(isopropoxycarbonyl)pyridin-1-ium br
Filed :
10-10-2023
Published :
N/A
Filed
1-(2-(Substituted phenyl)-2-oxoethyl)-4-methylpyridin-1-ium bromide as anti-tubercular agents
Katharigatta N. Venugopala
Pran Kishore Deb Mohamed A. Morsy
Bandar E. Aldhubiab
Sandeep Chandrashekharappa
Melendran Pillay
Chemical Sciences
Application No. :
18377407
Filed :
06-10-2023
Published :
N/A
Filed
(6-Methyl-4-substitutedphenyl-2-oxo/thioxo-1,2,3,4-tetrahydropyrimidin-5-yl)(piperidin-1-yl)methanones as anti-tubercular agents
Katharigatta N. Venugopala
Mohamed A. Morsy
Keshab M. Bairagi
Susanta K. Nayak
Melendran Pillay
Pran Kishore Deb
Sandeep Chandrashekharappa
Osama I. Alwassil
Chemical Sciences
Application No. :
18367645
Filed :
13-09-2023
Published :
N/A
Filed
(6-Methyl-4-substitutedphenyl-2-oxo/thioxo-1,2,3,4-tetrahydropyrimidin-5-yl)(piperidin-1-yl)methanones as anti-tubercular agents
Katharigatta N. Venugopala
Mohamed A. Morsy
Keshab M. Bairagi
Susanta K. Nayak
Melendran Pillay
Pran Kishore Deb
Sandeep Chandrashekharappa
Osama I. Alwassil
Chemical Sciences
Application No. :
18367635
Filed :
13-09-2023
Published :
N/A
Filed
Substituted 7-methyl quinoline derivatives as anti-tubercular agents.
Katharigatta N. Venugopala
Pran Kishore Deb
Melendran Pillay
Vijaykumar Uppar
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Sandeep Chandrashekharappa
Basavaraj Padmashali.
Chemical Sciences
Application No. :
18240256
Filed :
30-08-2023
Published :
N/A
Filed
Ethyl 2-substitued-1-(substitutedbenzoyl)-7-methylpyrrolo[1,2-a]quinoline-3-carboxylates as anti-tubercular agents.
Katharigatta N. Venugopala
Pran Kishore Deb
Melendran Pillay
Sandeep Chandrashekharappa
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Christophe Tratrat
Sheena Shashikanth
Vijaykumar Uppar
Basavaraj Padmashali.
Chemical Sciences
Application No. :
18237273
Filed :
23-08-2023
Published :
N/A
Filed
Ethyl 2-substitued-1-(substitutedbenzoyl)-7-methylpyrrolo[1,2-a]quinoline-3-carboxylates as anti-tubercular agents.
Katharigatta N. Venugopala
Pran Kishore Deb
Melendran Pillay
Sandeep Chandrashekharappa
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Christophe Tratrat
Sheena Shashikanth
Vijaykumar Uppar
Basavaraj Padmashali.
Chemical Sciences
Patent No. :
US Patent 11,845,746, 2023
Filed :
23-08-2023
Published :
19-12-2023
Granted
1-Substitutedbenzoyl-4-bromopyrrolo[1,2-a]quinoline-3-carboxylate derivatives as anti-tubercular agents
Katharigatta N. Venugopala
Pran Kishore Deb
Melendran Pillay
Sandeep Chandrashekharappa
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Vijaykumar Uppar
Raghu Prasad Mailavaram
Basavaraj Padmashali.
Chemical Sciences
Application No. :
18236237
Filed :
21-08-2023
Published :
N/A
Filed
Adenosine receptor activity of methyl/ethyl 3-(substituted benzoyl)-6,8-dimethylindolizine-2-substituted-1-carboxylates
Katharigatta N. Venugopala
Buccioni Michela
Gabriella Marucci
Pran Kishore Deb
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Sandeep Chandrashekharappa
Sheena Shashikanth.
Chemical Sciences
Application No. :
18230585
Filed :
08-08-2023
Published :
N/A
Filed
Novel substituted phenyl quinolin-1-ium bromide derivative as antitubercular agents.
Katharigatta N. Venugopala
Pran Kishore Deb
Melendran Pillay
Sandeep Chandrashekharappa
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Christophe Tratrat
Sheena Shashikanth
Chemical Sciences
Application No. :
18229825
Filed :
03-08-2023
Published :
N/A
Filed
7-Isopropyl 1-ethyl/methyl 3-(substituted benzoyl)-2-substituted indolizine-1,7-dicarboxylates as anti-tubercular agents
Katharigatta N. Venugopala
Bandar E. Aldhubiab
Mohamed A. Morsy
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Christophe Tratrat
Sandeep Chandrashekharappa
Melendran Pillay
Pran Kishore Deb
Sheena Shashikanth
Chemical Sciences
Application No. :
18191407
Filed :
30-03-2023
Published :
N/A
Filed
ANTI-TB NAPHTHYRIDINE DERIVATIVES AND THEIR SYNTHESIS THEREOF
Ningegowda
Raghu; Savitha H S
Neethu Patil; Chandrashekharappa
Sandeep
Chemical Sciences
Patent No. :
202341021764
Filed :
26-03-2023
Published :
31-03-2023
Filed
METHOD FOR SYNTHESIS OF CHRYSIN, TECTOCHRYSIN AND THEIR DERIVATIVES THEREOF FOR USE IN PHARMACEUTICAL APPLICATIONS
Niper Raebareli
Chemical Sciences
Patent No. :
202211047585
Filed :
22-08-2022
Published :
N/A
Filed
Antitubercular compounds
Katharigatta N Venugopala
Mahesh Attimarad
Anroop B Nair
Nagaraja Sreeharsha
Mohamed A Morsy
Sandeep Chandrashekharappa
Melendran Pillay
Pran Kishore Deb
-
Patent No. :
11530217
Filed :
29-06-2022
Published :
20-12-2022
Published
Compositions, materials, and methods for deactivating toxic agents;
InStem Bangalore
-
Patent No. :
IN 202142053063 A
Filed :
18-11-2021
Published :
10-12-2021
Published
N-(4-fluorophenyl)-5-phenyl-[1,2,4] triazolo [1,5-a] pyridine-2-carboxamide derivatives and their synthesis thereof
Ningegowda
Raghu; Banuprakash
Govindappa; Chandrashekharappa
Sandeep
Chemical Sciences
Patent No. :
WO 2021161084 A1
Filed :
19-08-2021
Published :
N/A
Published
Synthesis and characterization of (s)-3-(5-fluoropyridin-2-yl)-5-(piperidin-3-yl)-1,2,4-oxadiazole derivatives and their secretary phospholipase a2 (spla2) inhibitor activity
Ranjith Siddaraj
Raghu Ningegowda
Govindappa Banuprakash
Sandeep Chandrashekharappa
-
Patent No. :
WO 2022069953
Filed :
27-03-2021
Published :
07-04-2022
Published
Urolithin a and derivatives thereof for use in therapy
Jala
Venkatakrishna Rao; Bodduluri
Haribabu; Singh
Rajbir; Vemula
Praveen Kumar; Chandrashekharappa
Sandeep; Hiwale
Ankita Arun
-
Patent No. :
IN 202017054042 A
Filed :
26-02-2021
Published :
N/A
Published
Synthesis and characterization of (s)-3-(5-fluoropyridin-2-yl)-5-(piperidin-3-yl)-1,2,4-oxadiazole derivatives and their secretary phospholipase a2 (spla2) inhibitor activity
Ranjith Siddaraj
Raghu Ningegowda
Govindappa Banuprakash
Sandeep Chandrashekharappa
-
Patent No. :
457614
Filed :
29-09-2020
Published :
23-04-2021
Published
Ethyl and dimethyl 1-benzoylpyrrolo [1,2-a] quinoline-3-carboxylate analog derivatives as antifungal and antibacterial agents
Basavaraj Padmashali
Vijayakumar Uppar
. Sandeep Chandrashekharappa
Kiran K. MudnakuduNagaraju
-
Patent No. :
394853
Filed :
12-08-2019
Published :
05-02-2021
Granted
Compounds, compositions, methods of using and methods for preparing comopunds
Jala VR
Bodduluri H
Singh R
Vemula PK
Chandrashekharappa S
Hiwale AA
-
Patent No. :
US 2021/0267932 A1
Filed :
14-05-2019
Published :
02-09-2021
Published
Compositions, materials, and methods for deactivating toxic agents
InStem Bangalore
-
Patent No. :
20419
Filed :
21-03-2019
Published :
N/A
Filed
Treatment of Tuberculosis
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Pillay Melendhran
Bharti Odhav
Mohanlall Viresh
Kasumbwe kabange
-
Patent No. :
ZA 2020003088 A
Filed :
19-03-2019
Published :
30-06-2021
Published
Eco-friendly synthesis of pyrrolo [1,2-a] quinoline-3-carboxylate derivatives & their study of antibacterial and antioxidant properties
Vijayakumar Uppar
Basavaraj Padmashali
Govindappa Banuprakash
and Sandeep Chandrashekharappa
Chemical Sciences
Patent No. :
418528
Filed :
12-02-2019
Published :
13-03-2020
Granted
N-(4-fluorophenyl)-5-phenyl-[1,2,4] triazolo [1,5-a] pyridine-2-carboxamide derivatives and their synthesis thereof
Raghu Ningegowda
Sandeep Chandrashekharappa
Govindappa Banuprakash
-
Patent No. :
399540
Filed :
21-01-2019
Published :
20-06-2022
Published
Novel Substituted Indolizine Scaffolds For MDR Strains OF Mycobacterium Tuberculosis, Synthetic Methodology And Chemical Structures Thereof
Sandeep Chandrashekharappa. Katharigatta N. Venugopala.
-
Patent No. :
IN 201941002546 A
Filed :
21-01-2019
Published :
03-04-2020
Published
Synthetic analogs of gut microbial metabolites for protection of endothelial and epithelial barriers and applications thereof
Jala VR
Bodduluri H
Singh R
Vemula PK
Chandrashekharappa S
Hiwale AA
-
Patent No. :
11202011261P
Filed :
15-05-2018
Published :
30-12-2020
Published
Urolithin a and derivatives thereof for use in therapy
InStem Bangalore
Chemical Sciences
Patent No. :
WO 2019222146
Filed :
14-03-2018
Published :
21-11-2019
Published
Compositions, materials, and methods for deactivating toxic agents
InStem Bangalore
Chemical Sciences
Patent No. :
WO 2019180653 A1
Filed :
13-02-2018
Published :
26-09-2019
Published
A conjugate, a composition, an article, processes of preparation and application thereof
InStem Bangalore
Chemical Sciences
Patent No. :
201841006678
Filed :
13-02-2018
Published :
27-09-2019
Published
Greener synthesis of indolizine compounds
Sandeep C
Basavaraj Padmashali and Rashmi S. Kulkarni
Chemical Sciences
Patent No. :
359559
Filed :
09-10-2015
Published :
17-03-2017
Granted